PQR514 is a potent PI3K inhibitor with anticancer activity. PQR514 is able to inhibit cancer cell proliferation. PQR514 showed significant antitumor activity in the OVCAR-3 xenograft model, with the required concentration being approximately one-eighth that of PQR309. PQR514 has good pharmacokinetic properties and minimal brain penetration, making it an optimized candidate compound for inhibiting systemic tumors[1].
Molekulargewicht:
394.38
Reinheit:
97.73
CAS Nummer:
[1927857-55-3]
Formel:
C16H20F2N8O2
Target-Kategorie:
PI3K
Anwendungsbeschreibung:
MCE Product type: Reference compound1
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