PROTAC MPS1 degrader 2

Artikelnummer: MCE-HY-168543
Artikelname: PROTAC MPS1 degrader 2
Artikelnummer: MCE-HY-168543
Hersteller Artikelnummer: HY-168543
Alternativnummer: MCE-HY-168543-5MG,MCE-HY-168543-50MG,MCE-HY-168543-10MG,MCE-HY-168543-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC MPS1 degrader 2 (Compound 15) is a potent degrader of monopolar spindle 1 (Mps1, TTK), AURKA and AURKB, with DC50s of 42.0, 2.1 and 154.0 nM, respectively. PROTAC MPS1 degrader 1 can be used for the research of acute myeloid leukemia. (Pink: ligand for target protein (HY-168545), Black: linker (HY-N0420), Blue: ligand for E3 ligase (HY-10984)[1].
Molekulargewicht: 847.90
Reinheit: 99.7800
Formel: C41H41N11O8S
Target-Kategorie: Aurora Kinase,Mps1,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound