(E/Z)-4-Hydroxytamoxifen, CAS [[68392-35-8]]

Produktübersicht

• Artikelname: (E/Z)-4-Hydroxytamoxifen, CAS [[68392-35-8]]
• Artikelnummer: MCE-HY-16950A
• Hersteller Artikelnummer: HY-16950A
• Alternativnummer: MCE-HY-16950A-50MG,MCE-HY-16950A-100MG,MCE-HY-16950A-10MMX1ML,MCE-HY-16950A-10MG,MCE-HY-16950A-5MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: Afimoxifene, 4-OHT

Produktbeschreibung

(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is a racemic compound of (Z)-4-Hydroxytamoxifen and (E)-4-Hydroxytamoxifen isomers. (E/Z)-4-Hydroxytamoxifen is a selective estrogen receptor modulator with mixed estrogenic and antiestrogenic activity, which is also an active metabolite of Tamoxifen (HY-13757A). (E/Z)-4-Hydroxytamoxifen is an agonist of the G protein-coupled estrogen receptor (GPER) with relatively low affinity (100-1000 nM). (E/Z)-4-Hydroxytamoxifen is promising for research of cyclical mastalgia, such as breast pain, tenderness, and nodularity[1][2][3][4].

Produkteigenschaften

• Molekulargewicht: 387.51
• Reinheit: 99.62
• CAS Nummer: [68392-35-8]
• Formel: C26H29NO2
• Target-Kategorie: Adhesion G Protein-coupled Receptors (AGPCRs),Drug Metabolite,Estrogen Receptor/ERR

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound