EN1441 is a covalent degrader targeting the androgen receptor (AR) with an EC50 value of 4.2 µM and its truncated variant AR-V7. EN1441 selectively and potently degrades both AR and AR-V7 in androgen-independent prostate cancer cells. EN1441 is promising for research of androgen-independent prostate cancers[1].
Molekulargewicht:
264.71
Reinheit:
99.67
CAS Nummer:
[2196448-47-0]
Formel:
C13H13ClN2O2
Target-Kategorie:
Androgen Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten