(E)-Belizatinib, CAS [[1388225-72-6]] Preis auf Anfrage

Produktübersicht

• Artikelname: (E)-Belizatinib, CAS [[1388225-72-6]] Preis auf Anfrage
• Artikelnummer: MCE-HY-17603A
• Hersteller Artikelnummer: HY-17603A
• Alternativnummer: MCE-HY-17603A-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: (E)-TSR-011

Produktbeschreibung

(E)-Belizatinib ((E)-TSR-011)) (compound 36), the (E)-isomer of Belizatinib (HY-17603), is a potent, selective and orally active anaplastic lymphoma kinase (ALK) Inhibitor with an enzymatic IC50 of 0.005 µM and a cellular IC50 of 0.048 µM. (E)-Belizatinib shows >61-fold selectivity over JAK2, SRC, and IGF1R. (E)-Belizatinib shows favorable potency and PK characteristics in rats and dogs. (E)-Belizatinib can be used for ALK-driven cancer research[1].

Produkteigenschaften

• Molekulargewicht: 577.73
• CAS Nummer: [1388225-72-6]
• Formel: C33H44FN5O3
• Target-Kategorie: Anaplastic lymphoma kinase (ALK)

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound