Naperiglipron, CAS [[2572566-11-9]]

Artikelnummer: MCE-HY-177295
Artikelname: Naperiglipron, CAS [[2572566-11-9]]
Artikelnummer: MCE-HY-177295
Hersteller Artikelnummer: HY-177295
Alternativnummer: MCE-HY-177295-10MMX1ML,MCE-HY-177295-5MG,MCE-HY-177295-100MG,MCE-HY-177295-10MG,MCE-HY-177295-50MG,MCE-HY-177295-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: LY3549492
Naperiglipron (LY3549492) (Example 2) is a Glucagon-like peptide 1 receptor (GLP-1R) agonist with an EC50 of 1.14 nM for hGLP-1R. Naperiglipron significantly decreases the level of blood glucose in GLP-1R knock-in mouse models. Naperiglipron inhibits PDE10A1 enzyme activity (IC50: 7.43 µM) with a weak hERG inhibitory activity. Naperiglipron can be used for type II diabetes mellitus (T2DM) and obesity research[1].
Molekulargewicht: 580.58
Reinheit: 99.43
CAS Nummer: [2572566-11-9]
Formel: C33H26F2N4O4
Target-Kategorie: GLP Receptor,Phosphodiesterase (PDE)
Anwendungsbeschreibung: MCE Product type: Reference compound