Dyrk1A-IN-16, CAS [[2805339-74-4]] Preis auf Anfrage

Artikelnummer: MCE-HY-179600
Artikelname: Dyrk1A-IN-16, CAS [[2805339-74-4]] Preis auf Anfrage
Artikelnummer: MCE-HY-179600
Hersteller Artikelnummer: HY-179600
Alternativnummer: MCE-HY-179600-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Dyrk1A-IN-16 is a selective, brain-penetrant and ATP-competitive Dyrk1A inhibitor with a IC50 of 53 nM. Dyrk1A-IN-16 displays high selectivity across a broad kinase panel (specific for DYRK kinases) with nanomolar potency. Dyrk1A-IN-16 impairs neurosphere self-renewal, cell invasion, and EGFR stability in vitro. Dyrk1A-IN-16 inhibits tumor growth and prolongs survival in vivo. Dyrk1A-IN-16 has potential for glioblastoma (GBM) research[1].
Molekulargewicht: 303.29
CAS Nummer: [2805339-74-4]
Formel: C14H9NO5S
Target-Kategorie: DYRK,EGFR
Anwendungsbeschreibung: MCE Product type: Reference compound