Pelanserin (Compound 1) is an orally active antihypertensive agent. Pelanserin is a potent 5-HT2 receptor antagonist. Pelanserin has the ability to block the activity of alpha-adrenergic receptor, with its ED50 being 0.03 µg/mL. Pelanserin has vasodilatory activity, with its ED100 being 5 µg. Pelanserin exhibits antihypertensive activity in hypertensive rats and renal hypertensive dog breeds. Pelanserin can be used for research on hypertension[1][2][3].
Molekulargewicht:
364.44
CAS Nummer:
[2208-51-7]
Formel:
C21H24N4O2
Target-Kategorie:
5-HT Receptor,Adrenergic Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
