Pelanserin (Compound 1) is an orally active antihypertensive agent. Pelanserin is a potent 5-HT2 receptor antagonist. Pelanserin has the ability to block the activity of alpha-adrenergic receptor, with its ED50 being 0.03 µg/mL. Pelanserin has vasodilatory activity, with its ED100 being 5 µg. Pelanserin exhibits antihypertensive activity in hypertensive rats and renal hypertensive dog breeds. Pelanserin can be used for research on hypertension[1][2][3].
Molecular Weight:
364.44
CAS Number:
[2208-51-7]
Formula:
C21H24N4O2
Target:
5-HT Receptor,Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound
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