Naldemedine (tosylate), CAS [[1345728-04-2]] Preis auf Anfrage

Produktübersicht

• Artikelname: Naldemedine (tosylate), CAS [[1345728-04-2]] Preis auf Anfrage
• Artikelnummer: MCE-HY-19627A
• Hersteller Artikelnummer: HY-19627A
• Alternativnummer: MCE-HY-19627A-25MG,MCE-HY-19627A-10MMX1ML,MCE-HY-19627A-10MG,MCE-HY-19627A-5MG,MCE-HY-19627A-50MG,MCE-HY-19627A-1MG,MCE-HY-19627A-100MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: S-297995 (tosylate)

Produktbeschreibung

Naldemedine (S-297995) tosylate is an orally active µ-opioid receptor antagonist (PAMORA)[1]. Naldemedine tosylate shows potent binding affinities (Ki=0.34, 0.43, 0.94 nM, respectively) and antagonist activities (IC50=25.57, 7.09, 16.1 nM, respectively) for recombinant human µ-, delta-, and kappa- opioid receptors[2]. Naldemedine can be used in opioid-induced constipation (OIC) research[2]. Naldemedine tosylate is predicted to bind to 3CLpro encoded by SARS-CoV2 genome[3].

Produkteigenschaften

• Molekulargewicht: 742.84
• Reinheit: 92.16
• CAS Nummer: [1345728-04-2]
• Formel: C39H42N4O9S
• Target-Kategorie: Opioid Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound