Naldemedine (tosylate), CAS [[1345728-04-2]] Preis auf Anfrage

Product Overview

• Article Name: Naldemedine (tosylate), CAS [[1345728-04-2]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-19627A
• Supplier Catalog Number: HY-19627A
• Alternative Catalog Number: MCE-HY-19627A-25MG,MCE-HY-19627A-10MMX1ML,MCE-HY-19627A-10MG,MCE-HY-19627A-5MG,MCE-HY-19627A-50MG,MCE-HY-19627A-1MG,MCE-HY-19627A-100MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: S-297995 (tosylate)

Product Description

Naldemedine (S-297995) tosylate is an orally active µ-opioid receptor antagonist (PAMORA)[1]. Naldemedine tosylate shows potent binding affinities (Ki=0.34, 0.43, 0.94 nM, respectively) and antagonist activities (IC50=25.57, 7.09, 16.1 nM, respectively) for recombinant human µ-, delta-, and kappa- opioid receptors[2]. Naldemedine can be used in opioid-induced constipation (OIC) research[2]. Naldemedine tosylate is predicted to bind to 3CLpro encoded by SARS-CoV2 genome[3].

Product Properties

• Molecular Weight: 742.84
• Purity: 92.16
• CAS Number: [1345728-04-2]
• Formula: C39H42N4O9S
• Target: Opioid Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound