KV2 channel inhibitor-1 is a selective KV2 channel inhibitor with IC50s of 0.2 µM and 0.41 µM for KV2.1 and KV2.2, respectively. KV2 channel inhibitor-1 possesses good selectivity over KV1.2 (IC50>10 µM). KV2 channel inhibitor-1 is >10-fold selective over NaV channels and other KV channels and displays weak activity on CaV channels[1].
Molekulargewicht:
396.89
Reinheit:
98.73
CAS Nummer:
[689297-68-5]
Formel:
C20H17ClN4OS
Target-Kategorie:
Potassium Channel
Anwendungsbeschreibung:
MCE Product type: Reference compound1
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