KV2 channel inhibitor-1 is a selective KV2 channel inhibitor with IC50s of 0.2 µM and 0.41 µM for KV2.1 and KV2.2, respectively. KV2 channel inhibitor-1 possesses good selectivity over KV1.2 (IC50>10 µM). KV2 channel inhibitor-1 is >10-fold selective over NaV channels and other KV channels and displays weak activity on CaV channels[1].
Molecular Weight:
396.89
Purity:
98.73
CAS Number:
[689297-68-5]
Formula:
C20H17ClN4OS
Target:
Potassium Channel
Application Notes:
MCE Product type: Reference compound
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