Safinamide, CAS [[133865-89-1]]

Artikelnummer: MCE-HY-70057
Artikelname: Safinamide, CAS [[133865-89-1]]
Artikelnummer: MCE-HY-70057
Hersteller Artikelnummer: HY-70057
Alternativnummer: MCE-HY-70057-5MG,MCE-HY-70057-10MG,MCE-HY-70057-100MG,MCE-HY-70057-50MG,MCE-HY-70057-25MG,MCE-HY-70057-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: FCE 26743, EMD 1195686
Safinamide is a potent, selective, and reversible monoamine oxidase B (MAO-B) inhibitor (IC50=0.098 µM) over MAO-A (IC50=580 µM)[1]. Safinamide also blocks sodium channels and modulates glutamate (Glu) release, showing a greater affinity at depolarized (IC50=8 µM) than at resting (IC50=262 µM) potentials. Safinamide has neuroprotective and neurorescuing effects and can be used for the study of parkinson disease, ischemia stroke etc.al[2][3].
Molekulargewicht: 302.34
Reinheit: 99.89
CAS Nummer: [133865-89-1]
Formel: C17H19FN2O2
Target-Kategorie: Monoamine Oxidase
Anwendungsbeschreibung: MCE Product type: Reference compound