Mambalgin 1 (TFA)

Artikelnummer: MCE-HY-P1441A
Artikelname: Mambalgin 1 (TFA)
Artikelnummer: MCE-HY-P1441A
Hersteller Artikelnummer: HY-P1441A
Alternativnummer: MCE-HY-P1441A-1G,MCE-HY-P1441A-500UG,MCE-HY-P1441A-100UG
Hersteller: MedchemExpress
Kategorie: Proteine/Peptide
Mambalgin 1 TFA is a selective ASIC1a inhibitor (IC50 values are 192 and 72 nM for human ASIC1a and ASIC1a/1b dimer, respectively). Mambalgin 1 TFA binds to closed/inactive channel. Mambalgin 1 TFA is selective for ASIC1a over ASIC2a, ASIC3, TRPV1, P2X2, 5-HT3, Nav1.8, Cav3.2 and Kv1.2 channels. Mambalgin 1 TFA increases latency of withdrawal response in mouse tail-flick and paw-flick tests.
Molekulargewicht: 6554.54 (free acid)
Reinheit: 95.72
Formel: C272H429N85O84S10.xC2HF3O2
Target-Kategorie: Sodium Channel
Anwendungsbeschreibung: MCE Product type: Peptides