Mambalgin 1 (TFA)

Product Overview

• Article Name: Mambalgin 1 (TFA)
• Biozol Catalog Number: MCE-HY-P1441A
• Supplier Catalog Number: HY-P1441A
• Alternative Catalog Number: MCE-HY-P1441A-1G,MCE-HY-P1441A-500UG,MCE-HY-P1441A-100UG
• Manufacturer: MedchemExpress
• Category: Proteine/Peptide

Product Description

Mambalgin 1 TFA is a selective ASIC1a inhibitor (IC50 values are 192 and 72 nM for human ASIC1a and ASIC1a/1b dimer, respectively). Mambalgin 1 TFA binds to closed/inactive channel. Mambalgin 1 TFA is selective for ASIC1a over ASIC2a, ASIC3, TRPV1, P2X2, 5-HT3, Nav1.8, Cav3.2 and Kv1.2 channels. Mambalgin 1 TFA increases latency of withdrawal response in mouse tail-flick and paw-flick tests.

Product Properties

• Molecular Weight: 6554.54 (free acid)
• Purity: 95.72
• Formula: C272H429N85O84S10.xC2HF3O2
• Target: Sodium Channel

Application Notes

• Application Notes: MCE Product type: Peptides