GpTx-1 (TFA)

Produktübersicht

• Artikelname: GpTx-1 (TFA)
• Artikelnummer: MCE-HY-P1681A
• Hersteller Artikelnummer: HY-P1681A
• Alternativnummer: MCE-HY-P1681A-100UG,MCE-HY-P1681A-5MG,MCE-HY-P1681A-500UG,MCE-HY-P1681A-1MG
• Hersteller: MedchemExpress
• Kategorie: Proteine/Peptide

Produktbeschreibung

GpTx-1 TFA is a peptide-based NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. GpTx-1 TFA demonstrates potent inhibitory activity against the NaV1.7 channel with an IC50 value of 10 nM, while exhibiting excellent selectivity for NaV1.4 (IC50 = 0.301 µM) and NaV1.5 (IC50 = 4.20 µM), showing >20-fold and >950-fold selectivity respectively[1].

Produkteigenschaften

• Molekulargewicht: 4073.82 (free base)
• Reinheit: 99.56
• Formel: C176H271N53O45S7.xC2HF3O2
• Target-Kategorie: Sodium Channel

Anwendungsbeschreibung

• Anwendungsbeschreibung: Peptides