PROTAC ERRalpha ligand 1, CAS [[1264754-13-3]]

Artikelnummer: MCE-HY-U00425
Artikelname: PROTAC ERRalpha ligand 1, CAS [[1264754-13-3]]
Artikelnummer: MCE-HY-U00425
Hersteller Artikelnummer: HY-U00425
Alternativnummer: MCE-HY-U00425-10MG,MCE-HY-U00425-100MG,MCE-HY-U00425-5MG,MCE-HY-U00425-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC ERRalpha ligand 1 is a PROTAC target protein ligand. PROTAC ERRalpha ligand 1 is an orally active ERRalpha inverse agonist with IC50 values of 0.6 µM for ERRalpha. PROTAC ERRalpha ligand 1 shows no significant activity against a panel of other nuclear receptors, including ERalphac, ERRgamma, ERbeta, PPARalpha, PPARgamma, PPARdelta, and RXRalpha. PROTAC ERRalpha ligand 1 can provide enhanced insulin sensitivity in vivo. PROTAC ERRalpha ligand 1 can be used for metabolic diseases research, such as type 2 diabetes and obesity[1].
Molekulargewicht: 420.36
Reinheit: 99.47
CAS Nummer: [1264754-13-3]
Formel: C19H11F3N2O4S
Target-Kategorie: Estrogen Receptor/ERR,Ligands for Target Protein for PROTAC
Anwendungsbeschreibung: MCE Product type: Reference compound