PROTAC ERRalpha ligand 1 is a PROTAC target protein ligand. PROTAC ERRalpha ligand 1 is an orally active ERRalpha inverse agonist with IC50 values of 0.6 µM for ERRalpha. PROTAC ERRalpha ligand 1 shows no significant activity against a panel of other nuclear receptors, including ERalphac, ERRgamma, ERbeta, PPARalpha, PPARgamma, PPARdelta, and RXRalpha. PROTAC ERRalpha ligand 1 can provide enhanced insulin sensitivity in vivo. PROTAC ERRalpha ligand 1 can be used for metabolic diseases research, such as type 2 diabetes and obesity[1].
Molecular Weight:
420.36
Purity:
99.47
CAS Number:
[1264754-13-3]
Formula:
C19H11F3N2O4S
Target:
Estrogen Receptor/ERR,Ligands for Target Protein for PROTAC
Application Notes:
MCE Product type: Reference compound
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