GNF4877, CAS [[2041073-22-5]]

Artikelnummer: TGM-T11447
Artikelname: GNF4877, CAS [[2041073-22-5]]
Artikelnummer: TGM-T11447
Hersteller Artikelnummer: T11447
Alternativnummer: TGM-T11447-1MG,TGM-T11447-5MG,TGM-T11447-10MG,TGM-T11447-25MG,TGM-T11447-50MG,TGM-T11447-100MG,TGM-T11447-200MG
Hersteller: TargetMol
Kategorie: Biochemikalien
GNF4877 is a small molecule inhibitor, a potent dual-specificity kinase inhibitor targeting DYRK1A (IC50=6 nM) and GSK3beta (IC50=16 nM). This compound promotes beta-cell proliferation by blocking NFATc nuclear export (EC50=0.66 µM for mouse R7T1 cells) and is primarily used for research on beta-cell regeneration related to diabetes.
Molekulargewicht: 494.52
Reinheit: 98.63%
CAS Nummer: [2041073-22-5]
Formel: C25H27FN6O4
Target-Kategorie: GSK-3|||DYRK
T11447