Gintemetostat, CAS [[2604513-16-6]]

Artikelnummer: TGM-T202312
Artikelname: Gintemetostat, CAS [[2604513-16-6]]
Artikelnummer: TGM-T202312
Hersteller Artikelnummer: T202312
Alternativnummer: TGM-T202312-2MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: NSD2-IN-1 , KTX1001 , KTX-1001
Gintemetostat (KTX-1001) is a potent and selective small molecule inhibitor of nuclear receptor-binding SET domain protein 2 (NSD2), exhibiting IC50 values ranging from 0.001 µM to 0.01 µM, and it belongs to the chemical class of piperidinyl-methyl-purineamine derivatives, with primary research applications in oncology for the treatment of NSD2-dysregulated cancers.
Molekulargewicht: 546.52
CAS Nummer: [2604513-16-6]
Formel: C25H26F4N8O2
Target-Kategorie: Histone Methyltransferase
T202312