Gintemetostat (KTX-1001) is a potent and selective small molecule inhibitor of nuclear receptor-binding SET domain protein 2 (NSD2), exhibiting IC50 values ranging from 0.001 µM to 0.01 µM, and it belongs to the chemical class of piperidinyl-methyl-purineamine derivatives, with primary research applications in oncology for the treatment of NSD2-dysregulated cancers.
Molecular Weight:
546.52
CAS Number:
[2604513-16-6]
Formula:
C25H26F4N8O2
Target:
Histone Methyltransferase
T202312
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