Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage
Artikelnummer:
TGM-T212099
Hersteller Artikelnummer:
T212099
Alternativnummer:
TGM-T212099-10MG,TGM-T212099-50MG
Hersteller:
TargetMol
Kategorie:
Biochemikalien
Dopamine D3 receptor antagonist-3 is a selective positive allosteric modulator-antagonist (PAM-antagonist) of the D3 dopamine receptor (D3R) that can cross the blood-brain barrier. It demonstrates antagonistic activity in D3R-mediated beta-arrestin recruitment assays with an IC50 of 2.5 µM and Kb of 0.49 µM, and in D3R-mediated Go-BRET assays with an IC50 of 0.34 µM. Dopamine D3 receptor antagonist-3 is applicable for the study of neuropsychiatric disorders, including substance use disorders.
Molekulargewicht:
485.86
CAS Nummer:
[2894793-37-2]
Formel:
C18H17ClF5N3O3S
Target-Kategorie:
Dopamine Receptor
T212099
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