Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage

Artikelnummer: TGM-T212099
Artikelname: Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage
Artikelnummer: TGM-T212099
Hersteller Artikelnummer: T212099
Alternativnummer: TGM-T212099-10MG,TGM-T212099-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Dopamine D3 receptor antagonist-3 is a selective positive allosteric modulator-antagonist (PAM-antagonist) of the D3 dopamine receptor (D3R) that can cross the blood-brain barrier. It demonstrates antagonistic activity in D3R-mediated beta-arrestin recruitment assays with an IC50 of 2.5 µM and Kb of 0.49 µM, and in D3R-mediated Go-BRET assays with an IC50 of 0.34 µM. Dopamine D3 receptor antagonist-3 is applicable for the study of neuropsychiatric disorders, including substance use disorders.
Molekulargewicht: 485.86
CAS Nummer: [2894793-37-2]
Formel: C18H17ClF5N3O3S
Target-Kategorie: Dopamine Receptor
T212099