Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage

Product Overview

• Article Name: Dopamine D3 receptor antagonist-3, CAS [[2894793-37-2]] Preis auf Anfrage
• Biozol Catalog Number: TGM-T212099
• Supplier Catalog Number: T212099
• Alternative Catalog Number: TGM-T212099-10MG,TGM-T212099-50MG
• Manufacturer: TargetMol
• Category: Biochemikalien

Product Description

Dopamine D3 receptor antagonist-3 is a selective positive allosteric modulator-antagonist (PAM-antagonist) of the D3 dopamine receptor (D3R) that can cross the blood-brain barrier. It demonstrates antagonistic activity in D3R-mediated beta-arrestin recruitment assays with an IC50 of 2.5 µM and Kb of 0.49 µM, and in D3R-mediated Go-BRET assays with an IC50 of 0.34 µM. Dopamine D3 receptor antagonist-3 is applicable for the study of neuropsychiatric disorders, including substance use disorders.

Product Properties

• Molecular Weight: 485.86
• CAS Number: [2894793-37-2]
• Formula: C18H17ClF5N3O3S
• Target: Dopamine Receptor

Images

T212099