PF-4981517, CAS [[1390637-82-7]]

Artikelnummer: TGM-T21548
Artikelname: PF-4981517, CAS [[1390637-82-7]]
Artikelnummer: TGM-T21548
Hersteller Artikelnummer: T21548
Alternativnummer: TGM-T21548-1MLX10MM(INDMSO), TGM-T21548-1MG, TGM-T21548-5MG, TGM-T21548-10MG, TGM-T21548-25MG, TGM-T21548-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: CYP3cide
PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4). The IC 50 values for CYP3A activity are 0.03 µM,17 µM, and 71 µM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.
Molekulargewicht: 456.59
Reinheit: 99.77%
CAS Nummer: [1390637-82-7]
Formel: C26H32N8
Target-Kategorie: Cytochromes P450
T21548