PF-4981517 (CYP3cide) is a efficient, specific and time-dependent inhibitor of cytochrome P4503A4 (CYP3A4). The IC 50 values for CYP3A activity are 0.03 µM,17 µM, and 71 µM for CYP3A4, CYP3A5, and CYP3A7, respectively. PF-4981517 is able to be used to distinguish the contributions of CYP3A4 versus CYP3A5 on drug Metabolism.
Molecular Weight:
456.59
Purity:
99.77%
CAS Number:
[1390637-82-7]
Formula:
C26H32N8
Target:
Cytochromes P450
T21548
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