TC-N 22A, CAS [[1314140-00-5]]

Artikelnummer: TGM-T23440
Artikelname: TC-N 22A, CAS [[1314140-00-5]]
Artikelnummer: TGM-T23440
Hersteller Artikelnummer: T23440
Alternativnummer: TGM-T23440-1MG,TGM-T23440-5MG,TGM-T23440-10MG,TGM-T23440-25MG,TGM-T23440-50MG,TGM-T23440-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier. EC50 expression of TC-N 22A in BHK cells expressing human mGlu4 was 9 nM. TC-N 22A showed very low activity against mGlu 1, 2, 3, 5, and 7 receptors in excitation and forward allosteric models (EC50 >10 µM). TC-N 22A can be used in the study of central nervous system diseases.
Molekulargewicht: 283.35
Reinheit: 99.95%
CAS Nummer: [1314140-00-5]
Formel: C14H13N5S
Target-Kategorie: GluR
T23440