PD 151746, CAS [[179461-52-0]]
Artikelnummer:
TGM-T2493
- Bilder (1)
| Artikelname: | PD 151746, CAS [[179461-52-0]] |
| Artikelnummer: | TGM-T2493 |
| Hersteller Artikelnummer: | T2493 |
| Alternativnummer: | TGM-T2493-1MLX10MM(INDMSO),TGM-T2493-5MG,TGM-T2493-10MG,TGM-T2493-25MG,TGM-T2493-50MG |
| Hersteller: | TargetMol |
| Kategorie: | Biochemikalien |
| PD151746 is a calpain inhibitor with a 20-fold selectivity for u-calpain (Ki = 0.26 0.03 µM) over m-calpain (Ki = 5.33 0.77 µM). Its IC50 values are 0.26 0.03 µM (Ki for µ-calpain) and 5.33 0.77 µM (Ki for m-calpain) [1]. In vitro, PD151746 targets calpain and reduces oxLDL-induced cytotoxicity [2]. |
| Molekulargewicht: | 237.25 |
| Reinheit: | 95% |
| CAS Nummer: | [179461-52-0] |
| Formel: | C11H8FNO2S |
| Target-Kategorie: | Proteasome|||Cysteine Protease |

