PD 151746, CAS [[179461-52-0]]

Catalog Number: TGM-T2493
Article Name: PD 151746, CAS [[179461-52-0]]
Biozol Catalog Number: TGM-T2493
Supplier Catalog Number: T2493
Alternative Catalog Number: TGM-T2493-1MLX10MM(INDMSO),TGM-T2493-5MG,TGM-T2493-10MG,TGM-T2493-25MG,TGM-T2493-50MG
Manufacturer: TargetMol
Category: Biochemikalien
PD151746 is a calpain inhibitor with a 20-fold selectivity for u-calpain (Ki = 0.26 0.03 µM) over m-calpain (Ki = 5.33 0.77 µM). Its IC50 values are 0.26 0.03 µM (Ki for µ-calpain) and 5.33 0.77 µM (Ki for m-calpain) [1]. In vitro, PD151746 targets calpain and reduces oxLDL-induced cytotoxicity [2].
Molecular Weight: 237.25
Purity: 95%
CAS Number: [179461-52-0]
Formula: C11H8FNO2S
Target: Proteasome|||Cysteine Protease
T2493