UR-7247, CAS [[177847-28-8]]

Artikelnummer: TGM-T29075
Artikelname: UR-7247, CAS [[177847-28-8]]
Artikelnummer: TGM-T29075
Hersteller Artikelnummer: T29075
Alternativnummer: TGM-T29075-1MG,TGM-T29075-5MG,TGM-T29075-10MG,TGM-T29075-25MG,TGM-T29075-50MG,TGM-T29075-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: UR7247
UR-7247 is a novel orally active angiotensin II subtype I (AT1) antagonist, demonstrating very long pharmacological effects. in vivo studies indicate no significant difference between 10 mg UR-7247 and 100 mg losartan four hours post-administration, while in vitro blockade with 100 mg losartan exceeds that observed with UR-7247, confirming UR-7247s extended plasma half-life potentially due to high-affinity protein binding, highlighting its long-lasting, well-tolerated AT1 receptor antagonism in healthy subjects.
Molekulargewicht: 430.5
Reinheit: 98.88%
CAS Nummer: [177847-28-8]
Formel: C24H26N6O2
Target-Kategorie: RAAS
T29075
T29075