PF-04577806, CAS [[1072100-81-2]]

Artikelnummer: TGM-T38462
Artikelname: PF-04577806, CAS [[1072100-81-2]]
Artikelnummer: TGM-T38462
Hersteller Artikelnummer: T38462
Alternativnummer: TGM-T38462-5MG
Hersteller: TargetMol
Kategorie: Biochemikalien
PF-04577806 is a potent, selective, and ATP-competitive inhibitor of protein kinase C (PKC), showing significant inhibitory activity against various PKC isoforms, including PKCalpha (IC50=2.4 nM), PKCbetaI (IC50=8.1 nM), PKCbetaII (IC50=6.9 nM), PKCgamma (IC50=45.9 nM), and PKCtheta (IC50=29.5 nM). Additionally, it can reverse retinal vascular leakage in diabetic rats.
Molekulargewicht: 495.628
CAS Nummer: [1072100-81-2]
Formel: C26H37N7O3
Target-Kategorie: Others|||PKC|||Phosphatase
T38462