Vepdegestrant, CAS [[2229711-68-4]]

Produktübersicht

• Artikelname: Vepdegestrant, CAS [[2229711-68-4]]
• Artikelnummer: TGM-T39710
• Hersteller Artikelnummer: T39710
• Alternativnummer: TGM-T39710-1MLX10MM(INDMSO),TGM-T39710-1MG,TGM-T39710-5MG,TGM-T39710-10MG,TGM-T39710-25MG,TGM-T39710-50MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: Vepdegestrant

Produktbeschreibung

Vepdegestrant (ARV-471) is a selective and highly potent estrogen receptor (ER, ESR1) PROTAC degrader with strong degrading activity against the ER protein. By directly degrading the ER protein rather than merely antagonizing its activity, vepdegestrant effectively inhibits the ER signaling pathway and demonstrates significant antitumor activity in ER-positive (ER) breast cancer, with a DC50 value of approximately 2 nM. It is particularly effective against tumors harboring ESR1 mutations.

Produkteigenschaften

• Molekulargewicht: 723.9
• Reinheit: 97.15%
• CAS Nummer: [2229711-68-4]
• Formel: C45H49N5O4
• Target-Kategorie: Estrogen Receptor/ERR|||PROTACs

Bilder

T39710