Obatoclax (GX15-070), a pan-BCL-2 family proteins inhibitor and BH3 mimetic, exhibits a binding affinity (K_i) of 220 nM for BCL-2. It promotes autophagy-dependent cell death and cyclin D1 degradation via the proteasome. Additionally, Obatoclax demonstrates anti-cancer properties and broad-spectrum antiparasitic activity.
Molekulargewicht:
317.38
Reinheit:
99.44%
CAS Nummer:
[803712-67-6]
Formel:
C20H19N3O
Target-Kategorie:
Parasite|||Bcl-2 Family|||Autophagy|||Others
T41278
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