A-674563 HCl (552325-73-2(free base)), CAS [[2070009-66-2]]

Artikelnummer: TGM-T4444
Artikelname: A-674563 HCl (552325-73-2(free base)), CAS [[2070009-66-2]]
Artikelnummer: TGM-T4444
Hersteller Artikelnummer: T4444
Alternativnummer: TGM-T4444-1MLX10MM(INDMSO),TGM-T4444-1MG,TGM-T4444-2MG,TGM-T4444-5MG,TGM-T4444-10MG,TGM-T4444-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
A-674563 is an orally available, ATP-competitive, and reversible inhibitor of Akt (Ki: 11 nM for Akt1) [1]. It exhibits inhibitory activity against PKA and Cdk2 (IC50: 16/46 nM) but is 10- to >1, 800-fold selective for Akt1 versus additional kinases in the CMGC, CAMK, and TK families [1].
Molekulargewicht: 394.9
Reinheit: 98%
CAS Nummer: [2070009-66-2]
Formel: C22H23ClN4O
Target-Kategorie: ERK|||Akt|||CDK|||PKC|||PKA
T4444