Alofanib, CAS [[1612888-66-0]]
Artikelnummer:
TGM-T5122
- Bilder (1)
| Artikelname: | Alofanib, CAS [[1612888-66-0]] |
| Artikelnummer: | TGM-T5122 |
| Hersteller Artikelnummer: | T5122 |
| Alternativnummer: | TGM-T5122-1MLX10MM(INDMSO),TGM-T5122-1MG,TGM-T5122-5MG,TGM-T5122-10MG,TGM-T5122-25MG,TGM-T5122-50MG,TGM-T5122-100MG |
| Hersteller: | TargetMol |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | RPT835 |
| Alofanib (RPT835) is a selective allosteric inhibitor of FGFR2 and has a dramatic inhibitory effect on FGF2-induced phosphorylation of FRS2a in KATO III cells (IC50 <10 nM). It has no direct effect on FGF2-dependent FGFR1 and FGFR3 phosphorylation levels in either cell lines and no effects on FGF2-FGFR2 binding. |
| Molekulargewicht: | 413.4 |
| Reinheit: | 99.81% |
| CAS Nummer: | [1612888-66-0] |
| Formel: | C19H15N3O6S |
| Target-Kategorie: | Apoptosis|||FGFR |

