PBRM1-BD2-IN-2, a selective and cell-active inhibitor of the polybromo-1 (PBRM1) bromodomain, exhibits binding affinity and inhibitory activity specifically targeting the PBRM1-BD2 domain, with Kd and IC50 values of 9.3 µM and 1.0 µM, respectively. This compound is utilized in cancer research.
Molekulargewicht:
311.14
Reinheit:
>99.99%
CAS Nummer:
[2819989-57-4]
Formel:
C14H9Cl2FN2O
Target-Kategorie:
Epigenetic Reader Domain
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten