TPBM, CAS [[6466-43-9]]

Artikelnummer: TGM-T60827
Artikelname: TPBM, CAS [[6466-43-9]]
Artikelnummer: TGM-T60827
Hersteller Artikelnummer: T60827
Alternativnummer: TGM-T60827-25MG,TGM-T60827-50MG,TGM-T60827-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
TPBM is a potent inhibitor of estrogen receptor alpha (ERalpha). The IC 50 value of TPBM for 17beta-estradiol (E2)-ERalpha is 9 µM. TPBM is not toxic to cells and reduces E2ERalpha recruitment to an endogenous estrogen-responsive gene. TPBM inhibits E2-dependent growth of ERalpha-positive cancer cells with an IC 50 value of 5 µM. TPBM does not affect estrogen-independent cell growth [1].
Molekulargewicht: 316.38
CAS Nummer: [6466-43-9]
Formel: C15H16N4O2S
Target-Kategorie: Estrogen Receptor/ERR|||Others
T60827