TPBM, CAS [[6466-43-9]]

Artikelnummer: TGM-T60827
Artikelname: TPBM, CAS [[6466-43-9]]
Artikelnummer: TGM-T60827
Hersteller Artikelnummer: T60827
Alternativnummer: TGM-T60827-1MLX10MM(INDMSO),TGM-T60827-1MG,TGM-T60827-5MG,TGM-T60827-10MG,TGM-T60827-25MG,TGM-T60827-50MG,TGM-T60827-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
TPBM is a potent estrogen receptor alpha (ERalpha) inhibitor with an IC50 value of 9 µM for disruption of 17beta-estradiol-ERalpha interaction, effectively reducing E2ERalpha recruitment to endogenous estrogen-responsive genes and inhibiting E2-dependent proliferation of ERalpha-positive cancer cells with an IC50 of 5 µM, while remaining non-toxic and not affecting estrogen-independent cell growth, making it a selective probe for ERalpha signaling research.
Molekulargewicht: 316.38
Reinheit: 99.64%
CAS Nummer: [6466-43-9]
Formel: C15H16N4O2S
Target-Kategorie: Estrogen Receptor/ERR
T60827
T60827