CCT128930 hydrochloride, CAS [[2453324-32-6]]

Artikelnummer: TGM-T6303L
Artikelname: CCT128930 hydrochloride, CAS [[2453324-32-6]]
Artikelnummer: TGM-T6303L
Hersteller Artikelnummer: T6303L
Alternativnummer: TGM-T6303L-1MLX10MM(INDMSO), TGM-T6303L-1MG, TGM-T6303L-5MG, TGM-T6303L-10MG, TGM-T6303L-25MG, TGM-T6303L-50MG, TGM-T6303L-100MG, TGM-T6303L-200MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: CCT128930 hydrochloride(885499-61-6 Free base)
CCT128930 hydrochloride (CCT128930 hydrochloride) is a potent and selective inhibitor of AKT with IC50 of 6 nM. CCT128930 hydrochloride induces cell cycle arrest, DNA damage, and autophagy. CCT128930 hydrochloride has 28-fold selectivity over the closely related PKA kinase (IC50: 168 nM) through the targeting of Met282 of AKT, as well as 20-fold selectivity over p70S6K (IC50: 120 nM).
Molekulargewicht: 378.3
Reinheit: 98.55%
CAS Nummer: [2453324-32-6]
Formel: C18H21Cl2N5
Target-Kategorie: Apoptosis|||Autophagy|||mTOR|||Akt|||PKA
T6303L