YM-202074, CAS [[299900-83-7]]

Artikelnummer: TGM-T69489
Artikelname: YM-202074, CAS [[299900-83-7]]
Artikelnummer: TGM-T69489
Hersteller Artikelnummer: T69489
Alternativnummer: TGM-T69489-25MG,TGM-T69489-50MG,TGM-T69489-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
YM-202074 is a high affinity, selective metabotropic glutamate receptor type 1 (mGlu1) antagonist. YM-202074 binds an allosteric site of the rat mGlu1 receptor with a Ki of 4.8 nM. It inhibits mGlu1-mediated inositol phosphates production (IC50 = 8.6 nM in rat cerebellar granule cells).
Molekulargewicht: 414.56
CAS Nummer: [299900-83-7]
Formel: C22H30N4O2S
Target-Kategorie: Others|||GluR
T69489