dBRD4-BD1, CAS [[2839318-19-1]]

Produktübersicht

• Artikelname: dBRD4-BD1, CAS [[2839318-19-1]]
• Artikelnummer: TGM-T69506
• Hersteller Artikelnummer: T69506
• Alternativnummer: TGM-T69506-25MG,TGM-T69506-50MG,TGM-T69506-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien

Produktbeschreibung

dBRD4-BD1 is a selective BRD4 bromodomain inhibitor. dBRD4-BD1 can selectively degrade BRD4 (DC50 = 280 nM). Notably, dBRD4-BD1 upregulates BRD2/3, a result not observed with degraders using pan-BET ligands. Designing BRD4 selectivity up front enables analysis of BRD4 biology without wider BET-inhibition and simplifies designing BRD4-selective heterobifunctional molecules, such as degraders with new E3 recruiting ligands or for additional probes beyond degraders.

Produkteigenschaften

• Molekulargewicht: 967
• CAS Nummer: [2839318-19-1]
• Formel: C50H53F3N8O9
• Target-Kategorie: Others|||Epigenetic Reader Domain|||PROTACs

Bilder

T69506