4-Me-PDTic HCl, CAS [[2209073-52-7]]

Produktübersicht

• Artikelname: 4-Me-PDTic HCl, CAS [[2209073-52-7]]
• Artikelnummer: TGM-T69798
• Hersteller Artikelnummer: T69798
• Alternativnummer: TGM-T69798-25MG,TGM-T69798-50MG,TGM-T69798-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien

Produktbeschreibung

4-Me-PDTic is a potent and selective Kappa Opioid Receptor Antagonist. 4-Me-PDTic had a Ke = 0.37 nM in a [35S]GTPgammaS binding assay and was 645- and >8100-fold selective for the kappa relative to the µ and delta opioid receptors, respectively. Calculated logBB and CNS (central nervous system) multiparameter optimization (MPO) and low molecular weight values all predict that 4-Me-PDTic will penetrate the brain and pharmacokinetic studies in rats shows that 4-Me-PDTic does indeed penetrate the brain.

Produkteigenschaften

• Molekulargewicht: 432.43
• CAS Nummer: [2209073-52-7]
• Formel: C21H35Cl2N3O2
• Target-Kategorie: Others

Bilder

T69798