Naldemedine tosylate, CAS [[1345728-04-2]]

Produktübersicht

• Artikelname: Naldemedine tosylate, CAS [[1345728-04-2]]
• Artikelnummer: TGM-T70929
• Hersteller Artikelnummer: T70929
• Alternativnummer: TGM-T70929-25MG, TGM-T70929-50MG, TGM-T70929-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: S-297995 tosylate

Produktbeschreibung

Naldemedine tosylate (S-297995) is an orally active µ-opioid receptor antagonist (PAMORA) with high binding affinities (K_i = 0.34, 0.43, 0.94 nM) and potent antagonist activities (IC_50 = 25.57, 7.09, 16.1 nM) towards human recombinant µ-, delta-, and kappa-opioid receptors, respectively. It is utilized in research on opioid-induced constipation (OIC) and is anticipated to interact with the 3CL proenzyme encoded by the SARS-CoV-2 genome.

Produkteigenschaften

• Molekulargewicht: 742.84
• CAS Nummer: [1345728-04-2]
• Formel: C39H42N4O9S
• Target-Kategorie: Others|||Opioid Receptor