AM-8508, CAS [[1338483-67-2]]

Artikelnummer: TGM-T70942
Artikelname: AM-8508, CAS [[1338483-67-2]]
Artikelnummer: TGM-T70942
Hersteller Artikelnummer: T70942
Alternativnummer: TGM-T70942-25MG,TGM-T70942-50MG,TGM-T70942-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
AM-8508 is a potent and selective PI3Kdelta inhibitor. AM-8508 showed good cellular potency (in vitro pAKT IC50 = 4.6 nM ). AM-8505 xhibited excellent HWB potency (HWB (pAKT) IC50 = 2.7 nM). AM-8508 inhibit KLH-specific antibodies in animal models, signifying its potential for the treatment of human inflammatory diseases. PI3Kalpha and PI3Kbeta are ubiquitously expressed and play a role in cell growth, division, and survival.
Molekulargewicht: 374.37
CAS Nummer: [1338483-67-2]
Formel: C19H15FN8
Target-Kategorie: Others
T70942