Theliatinib tartrate, CAS [[2413487-72-4]]

Artikelnummer: TGM-T72431
Artikelname: Theliatinib tartrate, CAS [[2413487-72-4]]
Artikelnummer: TGM-T72431
Hersteller Artikelnummer: T72431
Alternativnummer: TGM-T72431-25MG,TGM-T72431-50MG,TGM-T72431-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: Xiliertinib tartrate , HMPL-309 tartrate , Xiliertinib tartrate , HMPL-309 tartrate
Theliatinib (Xiliertinib) tartrate is a potent and highly selective EGFR inhibitor with ATP-competitive and orally active properties, showing a K_i of 0.05 nM and an IC_50 of 3 nM for EGFR, and an IC_50 of 22 nM for the EGFR T790M/L858R mutant, with over 50-fold selectivity for EGFR compared to other kinases.
Molekulargewicht: 592.6
CAS Nummer: [2413487-72-4]
Formel: C29H32N6O8
Target-Kategorie: EGFR|||Others
T72431