Theliatinib tartrate, CAS [[2413487-72-4]]

Product Overview

• Article Name: Theliatinib tartrate, CAS [[2413487-72-4]]
• Biozol Catalog Number: TGM-T72431
• Supplier Catalog Number: T72431
• Alternative Catalog Number: TGM-T72431-25MG,TGM-T72431-50MG,TGM-T72431-100MG
• Manufacturer: TargetMol
• Category: Biochemikalien
• Alternative Names: Xiliertinib tartrate , HMPL-309 tartrate , Xiliertinib tartrate , HMPL-309 tartrate

Product Description

Theliatinib (Xiliertinib) tartrate is a potent and highly selective EGFR inhibitor with ATP-competitive and orally active properties, showing a K_i of 0.05 nM and an IC_50 of 3 nM for EGFR, and an IC_50 of 22 nM for the EGFR T790M/L858R mutant, with over 50-fold selectivity for EGFR compared to other kinases.

Product Properties

• Molecular Weight: 592.6
• CAS Number: [2413487-72-4]
• Formula: C29H32N6O8
• Target: EGFR|||Others

Images

T72431