(S,R,S)-AHPC-Me, CAS [[1948273-02-6]]
Artikelnummer:
TGM-T7752
- Bilder (1)
| Artikelname: | (S,R,S)-AHPC-Me, CAS [[1948273-02-6]] |
| Artikelnummer: | TGM-T7752 |
| Hersteller Artikelnummer: | T7752 |
| Alternativnummer: | TGM-T7752-25MG,TGM-T7752-50MG,TGM-T7752-100MG |
| Hersteller: | TargetMol |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | VHL ligand 2 , E3 ligase Ligand 1A |
| (S,R,S)-AHPC-Me (E3 ligase Ligand 1A) (VHL ligand 2) is an (S,R,S)-AHPC-based VHL ligand used to recruit the von Hippel-Lindau (VHL) protein. It is utilized in the synthesis of ARV-771, a VHL E3 ligase-based BET PROTAC degrader that effectively degrades BET proteins in castration-resistant prostate cancer (CRPC) cells with a DC50 <1 nM. |
| Molekulargewicht: | 444.59 |
| Reinheit: | 99.86% |
| CAS Nummer: | [1948273-02-6] |
| Formel: | C23H32N4O3S |
| Target-Kategorie: | E3 Ligase Ligand-Linker Conjugates|||Ligands for E3 Ligase |

