DQP-997-74, CAS [[2377187-09-0]] Preis auf Anfrage

Produktübersicht

• Artikelname: DQP-997-74, CAS [[2377187-09-0]] Preis auf Anfrage
• Artikelnummer: TGM-T82528
• Hersteller Artikelnummer: T82528
• Alternativnummer: TGM-T82528-5MG,TGM-T82528-50MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien

Produktbeschreibung

Dihydroquinoline-pyrazoline DQP-997-74 (compound 2i) is a selective N-methyl-d-aspartate receptor (NMDAR) inhibitor that preferentially targets GluN2C/D subunits, with IC50 values of 0.069 µM and 0.035 µM, respectively, and possesses blood-brain barrier permeability. It enhances its inhibitory potency in a time-dependent manner when combined with the agonist glutamate, reducing epileptogenic events in a murine model of tuberous sclerosis complex (TSC)-induced epilepsy. DQP-997-74 is potentially applicable for the study of NMDAR-related neurological diseases [1].

Produkteigenschaften

• Molekulargewicht: 570.37
• CAS Nummer: [2377187-09-0]
• Formel: C28H19Cl2F2N3O4
• Target-Kategorie: Others|||iGluR

Bilder

T82528