CAN508, CAS [[140651-18-9]]

Artikelnummer: TGM-T8796
Artikelname: CAN508, CAS [[140651-18-9]]
Artikelnummer: TGM-T8796
Hersteller Artikelnummer: T8796
Alternativnummer: TGM-T8796-1MLX10MM(INDMSO),TGM-T8796-5MG,TGM-T8796-10MG,TGM-T8796-25MG,TGM-T8796-50MG,TGM-T8796-100MG,TGM-T8796-200MG
Hersteller: TargetMol
Kategorie: Biochemikalien
CAN508 is a potent ATP-competitive CDK9/cyclin T1 inhibitor with an IC50 of 0.35 µM. It also competitively inhibits Cdk2-cyclin E with respect to ATP, with Ki and IC50 values of 13.3 µM and 20 µM, respectively. CAN508 exhibits a 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes. [Antitumor activity.]
Molekulargewicht: 218.22
Reinheit: 98.65%
CAS Nummer: [140651-18-9]
Formel: C9H10N6O
Target-Kategorie: CDK
T8796