DFPQ, CAS [[911678-60-9]]

Artikelnummer: TGM-T87969
Artikelname: DFPQ, CAS [[911678-60-9]]
Artikelnummer: TGM-T87969
Hersteller Artikelnummer: T87969
Alternativnummer: TGM-T87969-25MG,TGM-T87969-50MG,TGM-T87969-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: AP-06-202
DFPQ is a powerful and selective beta-arrestin-biased negative allosteric modulator(NAM) targeting the beta2-adrenergic receptor. It specifically inhibits the interaction of beta-arrestin with beta2AR without altering beta-agonist-induced cAMP production. Additionally, DFPQ reduces functional desensitization of the beta2AR in airway smooth muscle, enhancing beta-agonists capacity to maintain bronchorelaxation and curbing cell migration during prolonged beta-agonist treatment.
Molekulargewicht: 354.4
CAS Nummer: [911678-60-9]
Formel: C20H20F2N4
T87969