G-5758, CAS [[2413455-99-7]]

Artikelnummer: TGM-T87983
Artikelname: G-5758, CAS [[2413455-99-7]]
Artikelnummer: TGM-T87983
Hersteller Artikelnummer: T87983
Alternativnummer: TGM-T87983-25MG,TGM-T87983-50MG,TGM-T87983-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
G-5758 is an orally active IRE1alpha inhibitor with an IC50 of 38 nM for XBP1s. It is used in studies involving multiple myeloma models [KMS-11], demonstrating good tolerance in rats at oral doses up to 500 mg/kg. G-5758 exhibits pharmacodynamic effects comparable to those induced by IRE1 knockdown.
Molekulargewicht: 588.58
CAS Nummer: [2413455-99-7]
Formel: C27H24F4N6O3S
Target-Kategorie: IRE1|||Liposome
T87983